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BPS Bioscience Inc.
中級(jí)會(huì)員 | 第3年

13829799985

當(dāng)前位置:BPS Bioscience Inc.>>Inhibitors / Activators>> 27020Panobinostat

Panobinostat

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產(chǎn)品型號(hào)27020

品       牌BPS Bioscience

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更新時(shí)間:2024-11-25 17:13:25瀏覽次數(shù):88次

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●Purchase●DescriptionPanobinostat,alsoknownasLBH-589,isahighlyactive,non-selectiveHDACinhibitor
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Description

Panobinostat, also known as LBH-589, is a highly active, non-selective HDAC inhibitor. IC50’s against HDAC s 1-9 range between 3 – 61 nM except for a slightly higher IC50 value of 248 nM for HDAC 8. Panobinostat inhibits tumor cell proliferation and induces apoptosis in breast cancer and T cell lymphoma cells. In addition to its tumor-suppressive activities, panobinostat induces histone H3K9 and histone H4K8 acetylation and decreases the level of c-Myc expression.

Synonyms
Faridak, LBH-589

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